SI-109
PG-20161-12068
Product information
- Catalog No.
- PG-20161-12068
- Product Name
- SI-109
- CAS No.
- 2429877-30-3
- Molecular Formula
- C40H44F2N7O9P
- Molecular Weight
- 835.8
- Purity
- Not specified
- Storage
- -20°C
- Shipping
- Ambient Temperature
- Documents
Missing values are marked “Not specified”. Request the technical information you need with your inquiry. For research use only.
Packaging & pricing
| Catalog No. | Packaging | Price (USD) | Stock | Inquiry action |
|---|---|---|---|---|
| PG-20161-12068 | 1 MG | USD 898 | In stock | |
| PG-20161-12068 | 5 MG | USD 2,991 | In stock | |
| PG-20161-12068 | 10 MG | USD 5,340 | In stock |
Prices are shown in USD. Final pricing, package availability and delivery are confirmed with your quotation.
General Information
- Product Name
- SI-109
- CAS No.
- 2429877-30-3
- Synonyms
- Not specified
- Molecular Formula
- C40H44F2N7O9P
- Molecular Weight
- 835.8
- Appearance
- Not specified
- Solubility
- Not specified
- Description
SI-109 is a STAT3 SH2 domain inhibitor with reported antitumor activity and an inhibition constant of Ki=9 nM. It inhibits STAT3 transcriptional activity with IC50=3 μM. SI-109 has been used together with an analog of the CRBN ligand lenalidomide to design the PROTAC STAT3 degrader SD-36.
It is cataloged in the STAT inhibitor group within PROTAC Linkers. Its molecular formula is C40H44F2N7O9P, and its listed molecular weight is 835.8.