PROTAC BRD4 Degrader-8

PG-20161-70938

Product information

Catalog No.
PG-20161-70938
Product Name
PROTAC BRD4 Degrader-8
CAS No.
3026420-38-9
Molecular Formula
C53H61F2N9O11S2
Molecular Weight
1102.3
Purity
Not specified
Storage
-20°C
Shipping
Ambient Temperature
Documents

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Packaging & pricing

Packaging and pricing for PG-20161-70938
Catalog No.PackagingPrice (USD)StockInquiry action
PG-20161-709381 MGUSD 866In stock
PG-20161-709385 MGUSD 2,984In stock

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General Information

Product Name
PROTAC BRD4 Degrader-8
CAS No.
3026420-38-9
Synonyms
Not specified
Molecular Formula
C53H61F2N9O11S2
Molecular Weight
1102.3
Appearance
Not specified
Solubility
Not specified
Description

PROTAC BRD4 Degrader-8 combines ligands for von Hippel-Lindau and BRD4 in a PROTAC construct. Reported IC50 values are 1.1 nM for BRD4 BD1 and 1.4 nM for BRD4 BD2, respectively. The compound has been reported to induce BRD4 protein degradation in PC3 prostate cancer cells. It is cataloged in the BRD4 ligand-1-based PROTAC category and has the molecular formula C53H61F2N9O11S2.