XMD 8-92
PG-20161-86573
Product information
- Catalog No.
- PG-20161-86573
- Product Name
- XMD 8-92
- CAS No.
- 1234480-50-2
- Molecular Formula
- C26H30N6O3
- Molecular Weight
- 474.6
- Purity
- Not specified
- Storage
- -20°C
- Shipping
- Ambient Temperature
- Documents
Missing values are marked “Not specified”. Request the technical information you need with your inquiry. For research use only.
Packaging & pricing
| Catalog No. | Packaging | Price (USD) | Stock | Inquiry action |
|---|---|---|---|---|
| PG-20161-86573 | 10 MG | USD 35 | In stock | |
| PG-20161-86573 | 25 MG | USD 72 | In stock | |
| PG-20161-86573 | 50 MG | USD 114 | In stock |
Prices are shown in USD. Final pricing, package availability and delivery are confirmed with your quotation.
General Information
- Product Name
- XMD 8-92
- CAS No.
- 1234480-50-2
- Synonyms
- Not specified
- Molecular Formula
- C26H30N6O3
- Molecular Weight
- 474.6
- Appearance
- Not specified
- Solubility
- Not specified
- Description
XMD 8-92 is an ERK5 (BMK1) inhibitor reported to block growth factor-induced cellular BMK1 activation, reduce BMK1 activity in in vitro kinase assays, and decrease BMK1-dependent MEF2C transactivation. It is cataloged in the BMK inhibitor section within the PROTAC Linkers collection.
Reported Kd values are 80 and 190 nM for ERK5 (BMK1) and BRD4, respectively. Additional reported targets include DCAMKL2, PLK4 and TNK1, with corresponding Kd values of 190, 600 and 890 nM. Its molecular formula is C26H30N6O3, and its molecular weight is 474.6.