GSK 6853
PG-20161-89324
Product information
- Catalog No.
- PG-20161-89324
- Product Name
- GSK 6853
- CAS No.
- 1910124-24-1
- Molecular Formula
- C22H27N5O3
- Molecular Weight
- 409.5
- Purity
- Not specified
- Storage
- -20°C
- Shipping
- Ambient Temperature
- Documents
Missing values are marked “Not specified”. Request the technical information you need with your inquiry. For research use only.
Packaging & pricing
| Catalog No. | Packaging | Price (USD) | Stock | Inquiry action |
|---|---|---|---|---|
| PG-20161-89324 | 10 MG | USD 80 | In stock | |
| PG-20161-89324 | 25 MG | USD 128 | In stock | |
| PG-20161-89324 | 50 MG | USD 206 | In stock |
Prices are shown in USD. Final pricing, package availability and delivery are confirmed with your quotation.
General Information
- Product Name
- GSK 6853
- CAS No.
- 1910124-24-1
- Synonyms
- Not specified
- Molecular Formula
- C22H27N5O3
- Molecular Weight
- 409.5
- Appearance
- Not specified
- Solubility
- Not specified
- Description
GSK 6853 is a potent, selective BRPF1 inhibitor listed in the BRPF inhibitor collection. Reported selectivity for BRPF1 over other bromodomains is >1600-fold. TR-FRET pIC50 values are 8.1 for BRPF1, 5.1/4.8 for BRPF2/3 and 4.7/<4.3 for BRD4 BD1/2.
The structural analog GSK9311 serves as an inactive control, with 125- and 185-fold reduced potency in cell-free and cell-based assays, respectively. GSK 6853 has the molecular formula C22H27N5O3 and a molecular weight of 409.5.