GSK 2801
PG-20161-10572
Product information
- Catalog No.
- PG-20161-10572
- Product Name
- GSK 2801
- CAS No.
- 1619994-68-1
- Molecular Formula
- C20H21NO4S
- Molecular Weight
- 371.5
- Purity
- Not specified
- Storage
- -20°C
- Shipping
- Ambient Temperature
- Documents
Missing values are marked “Not specified”. Request the technical information you need with your inquiry. For research use only.
Packaging & pricing
| Catalog No. | Packaging | Price (USD) | Stock | Inquiry action |
|---|---|---|---|---|
| PG-20161-10572 | 10 MG | USD 25 | In stock | |
| PG-20161-10572 | 25 MG | USD 59 | In stock |
Prices are shown in USD. Final pricing, package availability and delivery are confirmed with your quotation.
General Information
- Product Name
- GSK 2801
- CAS No.
- 1619994-68-1
- Synonyms
- Not specified
- Molecular Formula
- C20H21NO4S
- Molecular Weight
- 371.5
- Appearance
- Not specified
- Solubility
- Not specified
- Description
GSK 2801 is a selective, cell-permeable inhibitor of the BAZ2 family of bromodomain-containing proteins. For BAZ2A and BAZ2B, respectively, the reported Kd values are 0.26 and 0.14 µM, with IC50 values of 0.40 and 0.43 μM.
No interaction is reported with the bromodomains of BRD4(BD1), CREBBP, TRIM24/TIF1α, PB1(BD5), PCAF, or ATAD2. The compound has molecular formula C20H21NO4S and molecular weight 371.5, with a specified storage temperature of -20°C.