GSK 5959

PG-20161-44980

Product information

Catalog No.
PG-20161-44980
Product Name
GSK 5959
CAS No.
901245-65-6
Molecular Formula
C22H26N4O3
Molecular Weight
394.5
Purity
Not specified
Storage
-20°C
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Ambient Temperature
Documents

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Packaging & pricing

Packaging and pricing for PG-20161-44980
Catalog No.PackagingPrice (USD)StockInquiry action
PG-20161-4498010 MGUSD 59In stock
PG-20161-4498025 MGUSD 88In stock

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General Information

Product Name
GSK 5959
CAS No.
901245-65-6
Synonyms
Not specified
Molecular Formula
C22H26N4O3
Molecular Weight
394.5
Appearance
Not specified
Solubility
Not specified
Description

GSK 5959 is a BRPF1 inhibitor with IC50 = 80 nM and >100-fold selectivity over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. It inhibits the interaction between BRPF1 and histone H3.3, a process involved in epigenetic regulation of gene expression. Listed in the BRPF inhibitor category, it has molecular formula C22H26N4O3 and a listed storage condition of -20°C.